Experiment 954966
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | BIAN,J: GHOSH,TK: WANG,JC: GILL,DL:. (1991). IDENTIFICATION OF INTRACELLULAR CALCIUM POLLS.. 266(14) |
| Amount utilized | |
| Compound isolated | |
| Disease | 75% OF TOTAL INTRACELLULAR ATP-DEPENDENT CALCIUM ACCUMULATION IS BLOCKED. THIS THAPSIGARGIN-RESPONSIVE POLL IS RELEASED BY INOSITOL TRIPHOSPHATE IN THE PRESENCE OF GTP. COMPOUND INHIBITS UPTAKE INTO TWO POOLS, ONE INOSITOL-TRIPHOSPHATE SENSITIVE, THE OTHER INSENSITIVE, AND CALCIUM FROM THE LATTER CAN BE TRANSFERRED TO THE FORMER BY GTP-DEPENDENT TRANSLOCASE. |
| Dose amount | 30.0 NANOMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | IC50 |