Experiment 955082
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | IV |
| Organism | Empty organism |
| Citation | SOLARY,E: VELAY,I: CHAUFFERT,B: BIDAN,JM: CAILLOT,D: DUMAS,M: GUY,H:. (1991). SUFFICIENT LEVELS OF QUININE IN THE SERUM CIRCUMVENT THE MULTIDRUG RESISTANCE OF THE HUMAN LEUKEMIC CELL LINE K562/ADM.. 68(8) |
| Amount utilized | |
| Compound isolated | |
| Disease | PATIENTW WITH REFRACTORY ACUTE MYELOBLASTIC LEUKEMIAS OR REFRACTORY MULTIPLE MEYLOMAS WERE GIVEN DOSES RANGING FROM 7 TO 30 MG/KG/DAY. SERUM LEVELS BETWEEN 8 AND 11 MG/L WERE ACHIEVED WITHIN 24 TO 36 HOURS. PATIENTS EXPERIENCED NO TOXICITIES. |
| Dose amount | VAR |
| Number | 5 |
| Qualitative result | ACTIVE |
| Animal | HUMAN ADULT |
| Dose expression | DOSE |