Experiment 955451

Compounds isolated

Details

PropertyValue
Pharmacology
OrganismEmpty organism
CitationREEN,RK: SINGH,J:. (1991). IN VITRO AND IN VIVO INHIBITION OF PULMONARY CYTOCHROME P450 ACTIVITIES BY PIPERINE, A MAJOR INGREDIENT OF PIPER SPECIES.. 29(6)
Amount utilized
Compound isolated
DiseaseARYLHYDROCARBON HYDROXYLASE AND 7-ETHOXYCOUMARIN DEETHYLASE WERE NONCOMPETITIVELY INHIBITED BY 41% AND 53% RESPECTIVELY, WITHIN ONE HR OF ADMINISTRATION OF CMPD. ACTIVITY OF FORMER ENZYME RETURNED TO NORMAL MORE QUICKLY.
Dose amount25.0 MG
Number3
Qualitative resultACTIVE
AnimalRAT
Per unitKG
Dose expressionDOSE