Experiment 955453
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Administration route | INTRAGASTRIC |
| Organism | Empty organism |
| Citation | REEN,RK: SINGH,J:. (1991). IN VITRO AND IN VIVO INHIBITION OF PULMONARY CYTOCHROME P450 ACTIVITIES BY PIPERINE, A MAJOR INGREDIENT OF PIPER SPECIES.. 29(6) |
| Amount utilized | |
| Compound isolated | |
| Disease | ARYLHYDROCARBON HYDROXYLASE AND 7-ETHOXYCOUMARIN DEETHYLASE WERE NONCOMPETITIVELY INHIBITED BY 40% AND 60% WITHIN 1.5 HR OF ADMINISTRATION OF FIRST DOSE OF CMPD. INHIBITION WAS MAINTAINED WITH DAILY DOSE FOR UP TO 7 DAYS. |
| Dose amount | 15.0 MG |
| Number | 5 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Per unit | KG |
| Dose expression | DOSE |