Experiment 955534
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | ARNOLD,RS: NEWTON,AC:. (1991). INHIBITION OF THE INSULIN RECEPTOR TYROSINE KINASE BY SPHINGOSINE.. 30(31) |
| Amount utilized | |
| Compound isolated | |
| Disease | AUTOPHOSPHORYLATION OF INSULIN RECEPTORS FROM RAT LIVER WAS INHIBITED TRITON X-100 MICELLES. THIS EFFECT WAS PREVENTED IF PHOSPHATIDYLSERINE (10 MOL%) WAS INCORPORATED INTO MICELLE. HOWEVER, IF MICELLE WAS MADE TO MIMIC COMPOSITION OF INNER LEAF OF ERYTHROCYTE MEMBRANE, THE INHIBITORY EFFEC TOF COMPOUND PERSISTED. |
| Dose amount | 145.0 MICROMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Dose expression | IC50 |