Experiment 956531
Worktypes
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | HSU,CYJ: PERSONS,PE: SPADA,AP: BEDNAR,RA: LEVITZKI,A: ZILBERSTEIN,A:. (1991). KINETIC ANALYSIS OF THE INHIBITION OF THE EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE BY LAVENDUSTIN-A AND ITS ANALOGUE.. 266(31) |
| Amount utilized | |
| Compound isolated | |
| Disease | CMPD IS BOTH A SLOW AND TIGHT BINDING INHIBITOR OF EPIDERMAL GROWTH FACTOR RECEPTOR TYROSINE KINASE. CMPD IS A HYPERBOLIC MIXED-TYPE INHIBITOR WITH RESPECT TO BOTH ATP AND PEPTIDE SUBSTRATE. |
| Dose amount | 4.0 MICROMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Dose expression | CONC USED |