Experiment 960226

Details

PropertyValue
Pharmacology
OrganismTripterygium wilfordii (CELASTRACEAE)
CitationYE,WH: TAO,XL: ZHANG,NZ:. (1990). MECHANISM OF TREATING RHEUMATOID ARTHRITIS WITH POLYGLYCOSIDES OF TRIPTERYGIUM WILFORDII HOOK (T-11). III. STUDY ON INHIBITORY EFFECT OF T-11 ON IN VITRO IG SECRETED BY PERIPHERAL BLOOD MONOCULEAR CELLS FROM NORMAL CONTROLS AND RHEUMATOID ARTHRITIS. 12(3)
Amount utilized
Compound isolated
DiseaseTHE VITRO EFFECTS OF A POLYGLYCOSIDE FRACTION (T-11) OF THE TITLE PLANT WERE STUDIED ON IMMUNGLOBULIN (IG) PRODUCTION BY PERIPHERAL BLOOD MONONUCLEAR CELLS (PB-MC) FROM 17 HEALTHY PERSONS AND 8 RHEUMATOID ARTHRITIS (RA) PATIENTS. PB-MC'S, MONOCYTES AND LYMPHOCYTES WERE TREATED SEPARATELY WITH DIFFERENT DOSES OF T-II FOR DIFFERENT PERIODS OF TIME. CELLS IN DIFFERENT COMBINATIONS WERE CULTURED FOR 2 WEEKS UNDER POKEWEED MITOGEN(PWM) STIMULATION AND THE IGG AND IGM CONTENT OF CULTURE SUPERNATANTS WERE DETERMINED USING THE DOUBLE ANTIBODY SOLID-PHASE IMMUNORADIOMETRIC ASSAY. THERE WAS NO DIFFERENCE IN THE INHIBITORY EFFECT OF T-II ON INVETRO IGM AND IGG PRODUCTION BY PB-MC'S EITHER BETWEEN THE TWO TYPES OF IG OF BETWEEN HEALTHY INDIVIDUALS AND RHEUMATOID ARTHRITIS PATIENTS. T-II ACTS BOTH ON MONOCYTES + LYMPHOCYTES, BUT MORE STRONGLY ON THE LATTER. RESULTS OF THIS STUDY CORRELATE WELL WITH THOSE OF CLINICAL TRIALS, SUGGESTING THAT THE THERAPEUTIC EFFECT OF T-II IS ASSOCIATED WITH ITS IMMUNOSUPPRESSIVE ACTIVITY.
Dose amount2-50 MCG
Number1
Qualitative resultACTIVE
Per unitML
Dose expressionCONC USED
ExtractCHROMATOGRAPHIC FRACTION