Experiment 968860
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | GRANT,S: BOISE,L: WESTIN,E: HOWE,C: PETTIT,GR: TURNER,A: MC CRADY,C:. (1991). IN VITRO EFFECTS OF BRYOSTATIN 1 ON THE METABOLISM AND CYTOTOXICITY OF 1-B-D-ARABINOFURANOSYLCYTOSINE IN HUMAN LEUKEMIA CELLS.. 42(4) |
| Amount utilized | |
| Compound isolated | |
| Disease | BRYOSTATIN 1 INCREASED THE METABOLISM OF 1-BETA-D-ARABINOFURANOSYL-CYTOSIN (ARA) TO ARA-CTP, THE CYTOTOXIC METABOLITE, 6-8X. BRYOSTATIN TREATMENT ALSO INCREASED THE INCORPORATION OF ARA-CTP INTO CELLULAR DNA. |
| Dose amount | 12.5 NANOMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | CELL CULTURE |
| Dose expression | CONC USED |