Experiment 972717
Compounds isolated
Details
| Property | Value |
|---|---|
| Pharmacology | |
| Organism | Empty organism |
| Citation | SATO,K: ISHIDA,Y: WAKAMATSU,K: KATO,R: HONDA,H: OHIZUMI,Y: NAKAMURA,H: OHYA,M: LANCELIN,JM: KOHDA,D: INAGAKI,F:. (1991). ACTIVE SITE OF MU-CONOTOXN GIIIA, A PEPTIDE BLOCKER OF MUSCLE SODIUM CHANNELS.. 266(26) |
| Amount utilized | |
| Compound isolated | |
| Disease | ELECTRICALLY-INDUCED TWITCH TENSION WAS MEASURED. EFFECT DEPENDS ON THE PRESENCE OF ARG AT THE 13TH POSITION OF MOLECULE. |
| Dose amount | 0.175 MICROMOLS |
| Number | 1 |
| Qualitative result | ACTIVE |
| Animal | RAT |
| Dose expression | IC50 |