Experiment 973819

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeIV
OrganismEmpty organism
CitationGRAHAM,MA: BISSETT,D: SETANOIANS,A: HAMILTON,T: KERR,DJ: HENRAR,R: KAYE,SB:. (1992). PRECLINICAL AND PHASE I STUDIES WITH RHIZOXIN TO APPLY A PHARMACOKINETICALLY GUIDED DOSE-ESCALATION SCHEME.. 87(7)
Amount utilized
Compound isolated
DiseaseDOSE WAS ESCALATED BY EXTENDED FACTOR-OF-TWO METHOD. SIDE EFFECTS WERE: WEIGHT LOSS, SLUGGISHNESS, ATAXIA, TRANSIENT HEMATOLOGIC CHANGES AND HEMATURIA. DIARRHEA OCCURRED AT DOSES GREATER THAN 9 MG/SQM.
Dose amount0.8 MG
Number2
Qualitative resultACTIVE
AnimalMOUSE
Per unitSQ M BODY SURFACE
Dose expressionDOSE