Experiment 996982

Details

PropertyValue
Pharmacology
Administration routeIP
OrganismEmpty organism
CitationHSU,B: CHEN,JT: YANG,JL: CHANG,SY: YUEH,HF: WANG,TW: CHOU,CH:. (1980). NEW RESULTS IN PHARMACOLOGIC RESEARCH OF SOME ANTICANCER AGENTS.. 1980()
Amount utilized
Compound isolated
DiseaseDISTRIBUTED IN MANY INTERNAL ORGANS 1 HOUR AFTER INJECTION.HIGHEST RADIOACTIVITY WAS IN KIDNEY,LIVER + SPLEEN.ACTIVITY WAS ALSO HIGH IN GASTRIC + INTESTINAL CONTENTS AND MAY BE RELATED TO EXCRETION THRU THE BILIARY TRACT. RADIOACTIVITY WAS HIGHER IN PLASMA THAN IN BLOOD CELLS.SOME RADIOACTIVITY WAS DETECTED IN THE BRAIN AND HEART. BIOLOGICAL HALF LIFE WAS 13 MINUTES. BLOOD LEVELS WERE LOWER THAN WITH HOMOHARRINGTONINE. 24 HOURS AFTER INJECTION 27.5% WAS FOUND IN THE URINE AND 11.2% IN FECES.
Dose amount1.0 MG
Number4
Qualitative resultACTIVE
AnimalMOUSE
Per unitKG
Dose expressionDOSE