Experiment 880360

Compounds isolated

Details

PropertyValue
Pharmacology
Administration routeIV INFUSION
OrganismEmpty organism
CitationDORR,FA: KUHN,JG: PHILLIPS,J: VON HOFF,DD:. (1988). PHASE I CLINICAL AND PHARMACOKINETIC INVESTIGATION OF DIDEMNIN B, A CYCLIC DEPSIPEPTIDE.. 24(11)
Amount utilized
Compound isolated
DiseaseFORTY-THREE PATIENTS WERE TESTED IN PHASE I STUDY. THE DOSE-LIMITING TOXICITY INCLUDED NAUSEA AND VOMITING. MILD HEPTOTOXICITY WAS OBSERVED WITH MILD ELEVATIONS OF TRANSAMINASES AND BILIRUBIN.
Dose amountVAR
Number1
Qualitative result.
AnimalHUMAN ADULT
Dose expressionDOSE