Citation 163284
HALL,IH: LIOU,YF: OKANO,M: LEE,KH:. (1982). ANTITUMOR AGENTS 46: IN VITRO EFFECTS OF ESTERS OF BRUSATOL,BISBRUSATOL,AND RELATED COMPOUNDS ON NUCLEIC ACID PROTEIN SYNTHESIS OF P-388 LYMPHOCYTIC LEUKEMIA CELLS.. 71()
Citation Details
| Title | ANTITUMOR AGENTS 46: IN VITRO EFFECTS OF ESTERS OF BRUSATOL,BISBRUSATOL,AND RELATED COMPOUNDS ON NUCLEIC ACID PROTEIN SYNTHESIS OF P-388 LYMPHOCYTIC LEUKEMIA CELLS. |
|---|---|
| Authors | HALL,IH: LIOU,YF: OKANO,M: LEE,KH: |
| Year | 1982 |
| Volume | 71 |
| Issue |
Summary
Year: 1982
Journal: Unknown
Organisms and Their Experiments (19)
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
WEAK ACTIVITY
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
ACTIVE
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 9 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
ACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
ACTIVE
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
ACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
ACTIVE
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
WEAK ACTIVITY
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
INACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
ACTIVE
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 9 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
INACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
WEAK ACTIVITY
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
WEAK ACTIVITY
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
WEAK ACTIVITY
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
ACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
ACTIN POLYMERIZATION INHIBITION
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
INACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
INACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
WEAK ACTIVITY
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
INACTIVE
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
INACTIVE
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 9 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
ACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
ACTIVE
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 2 |
RNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 3 |
PROTEIN SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
DNA POLYMERASE INHIBITION
|
INACTIVE
|
||
| 5 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
WEAK ACTIVITY
|
||
| 6 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 7 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
WEAK ACTIVITY
|
||
| 8 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 9 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 10 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
INACTIVE
|
||
| 11 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 12 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
ACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
ACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
ACTIVE
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
ACTIN POLYMERIZATION INHIBITION
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
ACTIVE
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
ACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
ACTIVE
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
ACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
ACTIVE
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
ACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
ACTIVE
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
INACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
WEAK ACTIVITY
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
INACTIVE
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
INACTIVE
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 9 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
INACTIVE
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
INACTIVE
|
||
| 3 |
DIHYDROFOLATE REDUCTASE INHIBITION
|
WEAK ACTIVITY
|
||
| 4 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
WEAK ACTIVITY
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 6 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 8 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 9 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
||
| 10 |
DNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 11 |
RNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 12 |
PROTEIN SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
INACTIVE
|
||
| 3 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
WEAK ACTIVITY
|
||
| 4 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 6 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
WEAK ACTIVITY
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 8 |
ANTITUMOR ACTIVITY
|
ACTIVE
|
||
| 9 |
DNA SYNTHESIS INHIBITION
|
ACTIVE
|
||
| 10 |
RNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 11 |
PROTEIN SYNTHESIS INHIBITION
|
ACTIVE
|
Unknown organism
| Experiment # | Pharmacology Type | Worktypes | Compound | Results |
|---|---|---|---|---|
| 1 |
DNA POLYMERASE INHIBITION
|
WEAK ACTIVITY
|
||
| 2 |
FORMIC ACID INCORPORATION INTO PURINES INHIBITION
|
INACTIVE
|
||
| 3 |
PROTEIN SYNTHESIS INHIBITION DURING ELONGATION PROCESS
|
WEAK ACTIVITY
|
||
| 4 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 4)
|
INACTIVE
|
||
| 5 |
SUCCINATE DEHYDROGENASE INHIBITION(STATE 3)
|
INACTIVE
|
||
| 6 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 4)
|
INACTIVE
|
||
| 7 |
ALPHA-KETOGLUTARATE DEHYDROGENASE INHIBITION(STATE 3)
|
WEAK ACTIVITY
|
||
| 8 |
ANTITUMOR ACTIVITY
|
INACTIVE
|
||
| 9 |
DNA SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|
||
| 10 |
RNA SYNTHESIS INHIBITION
|
INACTIVE
|
||
| 11 |
PROTEIN SYNTHESIS INHIBITION
|
WEAK ACTIVITY
|